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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50149599'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Warwick

Curated by ChEMBL
LigandPNGBDBM50149599(CHEMBL3770310)
Affinity DataIC50:  6.20nMAssay Description:Agonist activity at human Adenosine A1 receptor transfected in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP production after 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Warwick

Curated by ChEMBL
LigandPNGBDBM50149599(CHEMBL3770310)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human Adenosine A1 receptor expressed in yeast cells coexpressed with chimeric GPA1/Galphai1 after 16 hrs by beta galactosidase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed