Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50113247'
TargetAdenosine receptor A2b(Homo sapiens (Human))
National Institute Of Diabetes & Digestive & Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50113247(3-Methyl-1-phenethyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataKi:  646nMAssay Description:Binding affinity at human Adenosine A2B receptor expressed in HEK-293 cells, using [125I]-ABOPX as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
National Institute Of Diabetes & Digestive & Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50113247(3-Methyl-1-phenethyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataKi:  5.53E+3nMAssay Description:Inhibition of [125I]-APOBX binding to rat Adenosine A2B receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed