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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50310924'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM50310924(CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...)
Affinity DataIC50:  6.70nMAssay Description:The use of a Fluorometric Imaging Plate Reader (FLIPR) to measure calcium flux in Adenosine-receptor expressing cells is a well-established technique...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAdenosine receptor A2b(Homo sapiens (Human))
Vernalis (R&D)

US Patent
LigandPNGBDBM50310924(CHEMBL1080421 | US9120807, 8 | {6-Ethylamino-2-[(p...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at human adeosine A2B receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed