Affinity DataKi: 26nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibitory activity against Adenosine A3 receptor by inhibiting specific [3H](R)-PIA binding to rat testis membranesMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from human A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Affinity for human Adenosine A3 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Inhibitory activity against Beta-glucosidase from E-coliMore data for this Ligand-Target Pair
Affinity DataKi: 97nMAssay Description:Binding affinity to rat adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity for Adenosine A3 receptor expressed in HEK 293 cells by displacing i[125I]-ABMECAMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity athuman Adenosine A3 receptor expressed in HEK 293 cells by [125I]AB-MECA displacement.More data for this Ligand-Target Pair
Affinity DataKi: 137nMAssay Description:Binding affinity towards Adenosine A3 receptor (W243 A mutant receptor)More data for this Ligand-Target Pair
Affinity DataKi: 142nMAssay Description:Binding affinity towards human Adenosine A3 receptor wild typeMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Binding affinity to human adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Tested for the binding affinity of A3 receptor by displacing N6-[[125I]-4-amino-3-iodobenzyl]-adenosine-5''-N-methyluronamide from membranes of CHO ...More data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Affinity to Adenosine A3 receptor of rat testis membrane using [3H](R)-PIA with 150 nM DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 274nMAssay Description:Displacement of [125I]- AB-MECA from rat adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 280nMAssay Description:Displacement of [3H]AB-MECA from human adenosine A3 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Displacement of [125I]-AB-MECA binding to human adenosine A3 receptor expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Displacement of [3H]AB-MECA from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 534nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from mouse A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 615nMAssay Description:Binding affinity towards Adenosine A3 receptor (H95A mutant receptor)More data for this Ligand-Target Pair
Affinity DataKi: 3.25E+3nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.86E+4nMAssay Description:Displacement of [3H]NECA from human recombinant adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.98E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, against human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 242nMAssay Description:Effect on forskolin-stimulated cyclic AMP production in intact chinese hamster ovary (CHO) cell expressing the human Adenosine A3 receptorMore data for this Ligand-Target Pair