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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50266649'
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50266649(CHEMBL4071338)
Affinity DataKi:  0.386nMAssay Description:Displacement of [3H]HEMADO from recombinant human adenosine A3A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50266649(CHEMBL4071338)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]NECA from recombinant rat adenosine A3 receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50266649(CHEMBL4071338)
Affinity DataEC50:  2.20nMAssay Description:Antagonist activity at recombinant human adenosine A3 receptor expressed in CHO cell membranes assessed as reversal of NECA-mediated inhibition of ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed