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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50392647'
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392647(CHEMBL2153559)
Affinity DataKi:  79.4nMAssay Description:Displacement of [3H]prazosin from human cloned alpha1D adrenoceptor expressed in CHO cell membranes after 30 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
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Curated by ChEMBL
LigandPNGBDBM50392647(CHEMBL2153559)
Affinity DataKd:  5.75nMAssay Description:Antagonist activity at alpha1D adrenoceptor in Sprague-Dawley rat thoracic aorta assessed as inhibition of noradrenaline-induced contractions after 3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed