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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50213028'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213028(CHEMBL74283)
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human Alpha-2A adrenergic receptor from cultured LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
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TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213028(CHEMBL74283)
Affinity DataEC50:  2.80nMAssay Description:Alpha-2A adrenergic receptor agonistic potency as inhibition of forskolin-stimulated synthesis of cyclic adenosine monophosphateMore data for this Ligand-Target Pair
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