Affinity DataKi: 46nMAssay Description:Displacement of [3H]RX821002 from human adrenergic alpha2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 76nMAssay Description:Agonist activity at human adrenergic alpha-2A receptor expressed in CHO cells assessed as extracellular acidification by cytosensor microphysiometryMore data for this Ligand-Target Pair
Affinity DataEC50: 76nMAssay Description:Agonist activity at human alpha2A adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair