Affinity DataKi: 44nMAssay Description:Displacement of rauwolscine from human Alpha-2C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity for human Alpha-2C adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosinMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Effective concentration at Alpha-2C adrenergic receptor from CHO-C4 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Alpha-2C adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair