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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50212997'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataKi:  25nMAssay Description:Binding affinity towards human Alpha-2C adrenergic receptor by the displacement of [3H]rauwolscineMore data for this Ligand-Target Pair
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TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50212997(CHEMBL310335)
Affinity DataEC50:  4.10nMAssay Description:Agonistic activity towards human Alpha-2C adrenergic receptor was measured as ability to inhibit forskolin-stimulated synthesis of cyclic adenosine m...More data for this Ligand-Target Pair
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