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Found 8 Enz. Inhib. hit(s) with Target = 'Alpha-2C adrenergic receptor' and Ligand = 'BDBM50218115'
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic Alpha-2C receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  257nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataKi:  363nMAssay Description:Displacement of [3H]RX 821002 from human adrenergic alpha-2c receptor expressed in CHO cells in presence of GppNHp/NaChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonistic potency at human adrenergic alpha2C receptor expressed in CHO cells assessed as forskolin-induced cAMP accumulationChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Universita` Di Camerino

Curated by ChEMBL
LigandPNGBDBM50218115((R)-2-[1-(3'-nitrobiphenyl-2-yloxy)ethyl]-4,5-dihy...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed