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Found 3 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50009575'
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0530nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from rat C-terminal EGFP-tagged APJ receptor expressed in CHO cell membranes after 3 hrs by Wallac gamma count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataIC50:  0.0250nMAssay Description:Displacement of [125I]-(Glp1,Nle11,Try14)apelin-13 from recombinant rat EGFP-fused apelin receptor expressed in CHO cell membrane measured after 3 hr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataEC50:  1.90nMAssay Description:Activation of recombinant human APJ expressed in rat Chem5 cells co-expressing Galpha15 by Calcium 6-QF dye based fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed