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Found 3 Enz. Inhib. hit(s) with Target = 'Arginase-1' and Ligand = 'BDBM290382'
TargetArginase-1(Homo sapiens (Human))
Mars

US Patent
LigandPNGBDBM290382((3R,4S)-3-amino-4-(3-boronopropyl)-1-(piperidin-3-...)
Affinity DataIC50:  125nMAssay Description:Inhibition of arginase I (ARG I) and arginase II (ARG II) by Formula I or Formula II compounds is followed spectrophotometrically at 530 nm. The comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetArginase-1(Homo sapiens (Human))
Mars

US Patent
LigandPNGBDBM290382((3R,4S)-3-amino-4-(3-boronopropyl)-1-(piperidin-3-...)
Affinity DataIC50: <250nMpH: 7.4 T: 2°CAssay Description:Inhibition of arginase I (ARG I) and arginase II (ARG II) by Formula I or Formula II compounds is followed spectrophotometrically at 530 nm. The comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetArginase-1(Homo sapiens (Human))
Mars

US Patent
LigandPNGBDBM290382((3R,4S)-3-amino-4-(3-boronopropyl)-1-(piperidin-3-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of arginase I (ARG I) and arginase II (ARG II) by Formula I or Formula II compounds is followed spectrophotometrically at 530 nm. The comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent