Found 5 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM25749' TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Affinity DataKd: 105nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
Affinity DataKd: 251nMAssay Description:Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparationMore data for this Ligand-Target Pair
Affinity DataKd: 724nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
Affinity DataKd: 174nMAssay Description:Antagonist activity of compound against Beta-1 adrenergic receptor in isolated guinea pig left atriaMore data for this Ligand-Target Pair
