Found 10 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM25753' TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Affinity DataKi: 170nMAssay Description:Displacement of [3H](-)-CGP12177 from human adrenergic beta1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.51E+3nMAssay Description:Displacement of [3H]-CGP12177 from human beta1 ADR expressed in HEK293T cell membranes after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Niigata College Of Pharmacy
Curated by PDSP Ki Database
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Displacement of [3H](-)CGP12177 from human recombinant Beta-1 adrenergic receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Displacement of [3H]CGP 12177 from human recombinant beta1 adrenergic receptor expressed in HEK293 cells measured after 60 mins by scintillation coun...More data for this Ligand-Target Pair
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of human alpha1 adrenoceptorMore data for this Ligand-Target Pair
Affinity DataKd: 219nMpH: 7.4 T: 2°CAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:In vitro beta-1 adrenergic receptor activity was determined via inhibition of the positive chronotropic actions of isoproterenol in isolated guinea p...More data for this Ligand-Target Pair
