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Found 2 Enz. Inhib. hit(s) with Target = 'Calcitonin gene-related peptide type 1 receptor' and Ligand = 'BDBM50173477'
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50173477((S)-N-[(R)-5-Amino-1-(4-pyridin-4-yl-piperazine-1-...)
Affinity DataIC50:  200nMpH: 7.4Assay Description:Affinity against human calcitonin gene related peptide receptor (1 uM) expressed in SK-N-MC cells using [125I]-CGRP as radioligand after 180 minutes ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcitonin gene-related peptide type 1 receptor(Rattus norvegicus)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50173477((S)-N-[(R)-5-Amino-1-(4-pyridin-4-yl-piperazine-1-...)
Affinity DataIC50:  7.05E+4nMpH: 7.4Assay Description:Affinity against calcitonin gene related peptide receptor (1 uM) in rat spleen using [125I]-CGRP as radioligand after 180 minutes of incubation at pH...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed