Affinity DataIC50: 0.100nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Inhibition of CDK2/cyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of CDK2 (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Binding constant for CDK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Binding constant for full-length CDK2More data for this Ligand-Target Pair
Affinity DataKd: 8.10nMAssay Description:Average Binding Constant for CDK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair