Found 43 Enz. Inhib. hit(s) with Target = 'D(1A) dopamine receptor' and Ligand = 'BDBM50001955' 
3D Structure (crystal)Affinity DataKi: 4.60nMAssay Description:Binding affinity to dopamine D1 receptor high binding site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]fenoldopam from Dopamine receptor D1 of rat striatum membranesMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor expressed in Ltk deficient fibroblast cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]SCH23390 from human D1 dopamine receptor expressed in Ltk fibroblast cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 182nMAssay Description:Binding Affinity was determined against Dopamine receptor D1 in rat striatal membranes using [3H]- SCH 23390 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]SCH-23390 from rat dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >221nMAssay Description:Tested for binding affinity towards rat striatal dopamine receptor D1 using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:In vitro displacement of [3H]-SCH-23,390 binding to rat striatal Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:In vitro affinity at Dopamine receptor D1 of rat striatum by [3H]-SCH-23,390 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 236nMAssay Description:Ability to displace [3H]-SCH-23,390 binding to rat striatal Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Dopamine receptor D1 affinity was tested in vitro against corpus striatum from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in L cells incubated for 60 mins by radio ligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Binding affinity to dopamine D1 receptor low binding site by radioligand displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 888nMAssay Description:In vitro binding affinity of the compound towards Dopamine receptor D1 by displacing [125I]-FISCH radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 238nMAssay Description:In vitro antagonist binding affinity was determined by displacing the [3H]-SCH- in rat striatal Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Compound was tested in vitro for binding affinity towards dopamine Dopamine receptor D1 in rat striatal membrane by using [3H]-SCH- 23390 as radiolig...More data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Inhibition of binding of [3H]SCH-23390 to Dopamine receptor D1 was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Affinity of the Compound for Dopamine D1 receptor in rat striatal membrane was determined in vitro using Dopamine Antagonist [3H]SCH-23390 as ligand.More data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Compound was evaluated in vitro for binding affinity to Dopamine receptor D1 in rat striatal membranes using D1 antagonist [3H]-SCH-23,390More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibitition of binding of [3H]-SCH-23,390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 432nMAssay Description:In vitro binding affinity towards rat Dopamine receptor D1 by [3H]-SCH-23,390 displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 444nMAssay Description:Binding affinity against Dopamine receptor D1 from rat brain corpus striatum membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Agonist activity at human recombinant dopamine D1 receptor expressed in CHO cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKd: 680nMAssay Description:Equilibrium dissociation constant against recombinant Dopamine receptor D1A expressed in COS7 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Agonist activity at C-terminal RLuc8-fused D1R (unknown origin) transfected in human HEK293T cells co-expressing N-terminal Venus-tagged beta-arresti...More data for this Ligand-Target Pair
Affinity DataEC50: 521nMAssay Description:Agonist activity at C-terminal RLuc8-fused D1R (unknown origin) transfected in human HEK293T cells co-expressing N-terminal Venus-tagged beta-arresti...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at D1R (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2 hrs by cAMP Glo...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Agonist activity at D1R (unknown origin) transfected in human HEK293T cells assessed as increase in cAMP accumulation incubated for 2 hrs by cAMP Glo...More data for this Ligand-Target Pair
