TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 18nMAssay Description:Displacement of [3H]7-OH-DPAT from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 35nMAssay Description:High binding affinity towards human dopamine receptor 2 (short) expressed in Chinese hamster ovary cells using [3H]spiperone (0.5 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2S expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 52nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 short receptor expressed in CHO cells; high binding affinityMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Effective concentration for [3H]thymidine uptake in growing CHO cells stably expressing the dopamine D4.2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 54nMAssay Description:Compound was evaluated for its ability to displace [3H]raclopride from dopamine receptor D2 in rat striatal homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:High inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2L expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cells; high binding affinityMore data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:In vitro binding affinity to displace [3H]spiperone from the cloned human dopamine receptor D2 long in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Mus musculus (Mouse))
Medical Research Service
Curated by PDSP Ki Database
Medical Research Service
Curated by PDSP Ki Database
Affinity DataKi: 260nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 870nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2short receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 950nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.19E+3nMAssay Description:Displacement of [3H]YM-09151-2 from human dopamine D2 receptor expressed in CHOp cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Tested for binding affinity against Dopamine receptor D2 like from bovine striatum membranes by using [3H]YM-09151-2 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 2.58E+3nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, low affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2S expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity (low) towards human dopamine receptor 2 short against radioligand [3H]spiperone, expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Binding affinity (low) towards human dopamine receptor 2 (long) against radioligand [3H]spiperone, expressed in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Low inhibition constant against [3H]-spiperone binding to human Dopamine receptor D2L expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 3.10E+4nMAssay Description:In vitro for its ability to displace [3H]- spiperone from cloned human dopamine D2 long receptor expressed in CHO cells; Low binding affinityMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]- -spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataIC50: 462nMT: 2°CAssay Description:Each medicament was dissolved in serum-free F12 culture medium containing 100 μM of IBMX. CHO cells which can stably express D2 receptor were pre-...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKd: 3.50E+3nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKd: 1.90E+3nMAssay Description:In vitro affinity at wild type Dopamine receptor D2 on C6 (glioma) cell membranes.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKd: 6.70E+3nMAssay Description:In vitro affinity at mutant D2 receptor (S194A) in C6 (glioma) cell membranes.More data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:Agonist activity at human dopamine D2 receptor expressed in CHOp cells assessed as stimulation of mitogenesis incubated for 24 hrs by [3H]thymidine i...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Dupont Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataEC50: 48nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair