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Found 2 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM205995'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chengdu Easton Pharmaceutical

US Patent
LigandPNGBDBM205995(US9255098, Ex. 1 | US9255098, Ex. 4)
Affinity DataIC50:  0.0500nMT: 2°CAssay Description:Gly-Pro-7-amido-4-methylcoumarin can be hydrolyzed by dipeptidyl peptidase IV (DPP-IV) at room temperature, to generate 7-amido-4-methyl coumarin, wh...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chengdu Easton Pharmaceutical

US Patent
LigandPNGBDBM205995(US9255098, Ex. 1 | US9255098, Ex. 4)
Affinity DataIC50:  0.0800nMT: 2°CAssay Description:Gly-Pro-7-amido-4-methylcoumarin can be hydrolyzed by dipeptidyl peptidase IV (DPP-IV) at room temperature, to generate 7-amido-4-methyl coumarin, wh...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent