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Found 1 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase Mdm2' and Ligand = 'BDBM31219'
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Schering-Plough Research Institute

LigandPNGBDBM31219(2-phenoxybenzoyltryptophan derivative, R4C1)
Affinity DataKi:  1.00E+4nM ΔG°:  -28.3kJ/molepH: 7.4 T: 2°CAssay Description:Ki values were determined from a competition experiment in which serial dilutions of inhibitor were added to compete against a fixed concentration (1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed