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Found 4 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase Mdm2' and Ligand = 'BDBM50436047'
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  916nMAssay Description:Displacement of fluorescent P4 peptide from recombinant human MDM2 (18 to 125) expressed in Escherichia coli BL21(DE3) RIL expression system after 30...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  916nMAssay Description:Binding affinity to human MDM2 by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  920nMAssay Description:Binding affinity to MDM2 (unknown origin) expressed in Escherichia coli BL21(DE3) after 30 mins by fluorescence polarization assay in presence of P4 ...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  920nMAssay Description:Competition binding affinity to MDM2 (unknown origin) using p53 mimicking peptide TSFAEYWNLLSP after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair