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Found 2 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 1' and Ligand = 'BDBM18125'
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University Of Groningen

Curated by ChEMBL
LigandPNGBDBM18125((2S)-2-aminobutanedioic acid | Aspartate | CHEMBL2...)
Affinity DataIC50:  9.33E+3nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed