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Found 1 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2' and Ligand = 'BDBM378893'
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM378893(5,8-dichloro-2-((7-methyl-5-oxo-5,6-dihydro-1H-pyr...)
Affinity DataIC50: <0.5nMAssay Description:Ten-point dose-response curves for a subset of compounds shown in Table 1 were determined using a TranscreenerŽ EPIGEN Methyltransferase HTS assay us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent