Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2' and Ligand = 'BDBM378911'
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM378911(7-((5,8-dichloro-7-(3,5-dimethylisoxazol-4-yl)-1-o...)
Affinity DataIC50:  3nMAssay Description:Ten-point dose-response curves for a subset of compounds shown in Table 1 were determined using a TranscreenerŽ EPIGEN Methyltransferase HTS assay us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent