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Found 1 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase EZH2' and Ligand = 'BDBM378913'
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Mirati Therapeutics

US Patent
LigandPNGBDBM378913(7-((5,8-dichloro-7-((1,1-dioxidothietan-3-yl)(meth...)
Affinity DataIC50:  2nMAssay Description:Ten-point dose-response curves for a subset of compounds shown in Table 1 were determined using a TranscreenerŽ EPIGEN Methyltransferase HTS assay us...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent