TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataKi: 197nMAssay Description:Binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataKi: 197nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]U-69593 as radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataKi: 298nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataKi: 1.13E+3nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+3nMAssay Description:Binding affinity against opioid receptor kappa 1 using [3H]- U-69,593 radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataIC50: 5.89E+3nMAssay Description:In vitro binding activity against opioid receptor kappa using [3H]-EKC as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Sri International
Curated by PDSP Ki Database
Sri International
Curated by PDSP Ki Database
Affinity DataIC50: 5.89E+3nMAssay Description:Compound was tested in vitro for binding affinity towards kappa opioid receptor by measuring displacement of [3H]-EKC from guinea pig brain membranesMore data for this Ligand-Target Pair