Affinity DataKi: 140nMAssay Description:Inhibition of [3H]diprenorphine binding to human KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Melbourne
Curated by PDSP Ki Database
The University Of Melbourne
Curated by PDSP Ki Database
Affinity DataKi: 163nMAssay Description:Inhibition of [3H]-U-69,593 binding to rat opioid receptor kappa 1 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 531nMAssay Description:Enhancement of [35S]GTPgammaS binding to human KOR expressed in CHO cellsMore data for this Ligand-Target Pair