Affinity DataKi: 2nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 137nMAssay Description:Agonist activity at kappa opioid receptor in human HEK293 cells assessed as stimulation of Galphai signaling by cAMP assayMore data for this Ligand-Target Pair