Affinity DataIC50: 9.08E+3nMAssay Description:Displacement of bis-ANS to recombinant human MD2 after 5 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKon: 0.703M-1s-1Assay Description:Binding affinity to MD2 (unknown origin) by SPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.25E+5nMAssay Description:In vitro inhibition against TXA2/PGH2 receptor using [3H]-SQ 29,548 as radioligand in human platelet membrane preparationMore data for this Ligand-Target Pair