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Found 1 Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 5A/5B' and Ligand = 'BDBM263991'
TargetLysine-specific demethylase 5A/5B(Homo sapiens (Human))
Celgene

Curated by ChEMBL
LigandPNGBDBM263991(2-{5-[(4-ethylbenzyl)oxy]- 1H-pyrazol-1-yl}pyridin...)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed