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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 5' and Ligand = 'BDBM463999'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM463999(US10787435, Example 002 | US11117891, Example 2 | ...)
Affinity DataIC50:  1.80nMAssay Description:The assay is done using an ADP-Glo™ Kinase Assay Kit (Promega, Catalog #V9102) according to the manufacturer's protocol with the following modifi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM463999(US10787435, Example 002 | US11117891, Example 2 | ...)
Affinity DataIC50: <50nMAssay Description:Reagents:Base Reaction Buffer: 20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM EGTA, 0.02% Brij35, 0.02 mg/ml BSA, 0.1 mM Na3VO4, 2 mM DTT, 1% DMSOCompound T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent