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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase kinase 2' and Ligand = 'BDBM51922'
LigandPNGBDBM51922(2-[4-(2,5-dimethylphenyl)-1-piperazinyl]-6,7-dimet...)
Affinity DataEC50:  3.89E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
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LigandPNGBDBM51922(2-[4-(2,5-dimethylphenyl)-1-piperazinyl]-6,7-dimet...)
Affinity DataEC50:  5.31E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03MH084830-01 Project Title: TR-FRET HTS Assay for Inhibitors of MEKK2-MEK5 PB1 Domain...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay