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Compile Data Set for Download or QSAR
maximum 50k data
Found
2
Enz. Inhib. hit(s) with Target = 'Monoglyceride lipase' and Ligand = 'BDBM474415'
Target
Monoglyceride lipase
(Homo sapiens (Human))
Pfizer
US Patent
Ligand
BDBM474415
(1-({[(3R)-3-(4-Fluoro-1H-pyrazol-1-yl)-1-oxa-8-aza...)
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Affinity Data
IC50: 121nM
Assay Description:
T = 30 minutes.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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Target
Monoglyceride lipase
(Homo sapiens (Human))
Pfizer
US Patent
Ligand
BDBM474415
(1-({[(3R)-3-(4-Fluoro-1H-pyrazol-1-yl)-1-oxa-8-aza...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.95E+3nM
Assay Description:
Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI