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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50083652'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50083652(CHEMBL112297 | Hexadecanoic acid (S)-2-benzyloxyca...)
Affinity DataKi:  0.229nMAssay Description:Ability to displace [3H]QNB from HM2 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50083652(CHEMBL112297 | Hexadecanoic acid (S)-2-benzyloxyca...)
Affinity DataKi:  0.229nMAssay Description:Binding of [3H]-QNB to HM2 receptor was evaluated by saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50083652(CHEMBL112297 | Hexadecanoic acid (S)-2-benzyloxyca...)
Affinity DataKi:  851nMAssay Description:Ability to displace [3H]QNB from HM2 receptor binding to acetylcholine was evaluated by ligand inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50083652(CHEMBL112297 | Hexadecanoic acid (S)-2-benzyloxyca...)
Affinity DataKd:  1.80nMAssay Description:Binding of [3H]QNB to HM2 receptor was evaluated by saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed