Found 4 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50212288'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair