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Found 2 Enz. Inhib. hit(s) with Target = 'PAS domain-containing serine/threonine-protein kinase' and Ligand = 'BDBM463535'
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix

US Patent
LigandPNGBDBM463535(2-(4-Cyanophenyl)-3-(isopropyl(methyl)amino)quinox...)
Affinity DataIC50: <1.00E+3nMAssay Description:Compound screening was done via the following method. 10 mM stock solution of test compound in DMSO was prepared by dissolving test compound in DMSO ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPAS domain-containing serine/threonine-protein kinase(Homo sapiens (Human))
Bioenergenix

US Patent
LigandPNGBDBM463535(2-(4-Cyanophenyl)-3-(isopropyl(methyl)amino)quinox...)
Affinity DataIC50: <1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent