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Found 2 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase FKBP1A' and Ligand = 'BDBM50240505'
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240505(CHEMBL4077559)
Affinity DataIC50:  11nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240505(CHEMBL4077559)
Affinity DataIC50:  824nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed