Found 2 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase FKBP1A' and Ligand = 'BDBM50240505'
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Amplyx Pharmaceuticals
Curated by ChEMBL
Amplyx Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Homo sapiens (Human))
Amplyx Pharmaceuticals
Curated by ChEMBL
Amplyx Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 824nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair