Found 6 Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor beta' and Ligand = 'BDBM50237710'
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged PDGFRbeta cytoplasmic domain (557 to 1106 residues) expressed in baculovirus expression system ...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 60nMAssay Description:Inhibition of human PDGFRbeta using poly[Glu:Tyr] (4:1) peptide substrateMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataIC50: 71nMAssay Description:Inhibition of PDGFRbeta autophosphorylation in human A31 cells by ELISAMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 16nMAssay Description:Binding affinity to human PDGFRbeataMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Genomics Institute Of The Novartis Research Foundation
Curated by PDSP Ki Database
Affinity DataKd: 73nMAssay Description:Binding constant for PDGFRB kinase domainMore data for this Ligand-Target Pair