Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM18660'
TargetProgesterone receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM18660((10S,11S,14S,15S)-14,15-dimethyl-14-propanoyltetra...)
Affinity DataIC50:  0.236nMAssay Description:Agonist activity at GAL4 DNA-binding domain fused PR (unknown origin) ligand binding domain expressed in UAS-bla HEK 293T cells assessed as beta-lact...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM18660((10S,11S,14S,15S)-14,15-dimethyl-14-propanoyltetra...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed