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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM50375442'
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375442(CHEMBL260764)
Affinity DataIC50:  0.600nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50375442(CHEMBL260764)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at human PRB expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed