Affinity DataIC50: 0.600nMAssay Description:Antagonist activity at human PRB expressed in CHO cells assessed as inhibition of Org 2058 induced-transactivationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.230nMAssay Description:Agonist activity at human PRB expressed in CHO cellsMore data for this Ligand-Target Pair