Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-7' and Ligand = 'BDBM50007195'
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  76nMAssay Description:Inhibition of caspase-like activity of human 20S proteasome using Ac-nLPnLD-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Hokkaido University

Curated by ChEMBL
LigandPNGBDBM50007195(CHEMBL3237866)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Ac-RLR-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed