Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Ras-related C3 botulinum toxin substrate 1' and Ligand = 'BDBM54709'
LigandPNGBDBM54709(1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...)
Affinity DataKi:  20nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54709(1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...)
Affinity DataKi:  300nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54709(1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...)
Affinity DataEC50:  257nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54709(1-[4-(4-bromophenyl)-1-piperazinyl]-3-[3-(4-methox...)
Affinity DataEC50:  3.26E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay