Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Replicase polyprotein 1ab' and Ligand = 'BDBM50458462'
TargetReplicase polyprotein 1ab(Middle East respiratory syndrome-related coronavir...)
Wichita State University

Curated by ChEMBL
LigandPNGBDBM50458462(CHEMBL4214066)
Affinity DataIC50:  600nMAssay Description:Inhibition of Middle East respiratory syndrome-related coronavirus 3CL protease using Dabcyl-KTSAVLQ/SGFRKME-Edans as substrate incubated for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Feline coronavirus (strain FIPV WSU-79/1146) (FCoV...)
Wichita State University

Curated by ChEMBL
LigandPNGBDBM50458462(CHEMBL4214066)
Affinity DataIC50:  800nMAssay Description:Inhibition of Feline infectious peritonitis virus 3CL protease using Dabcyl-KTSAVLQ/SGFRKME-Edans as substrate incubated for 30 mins followed by subs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReplicase polyprotein 1ab(Human SARS coronavirus (SARS-CoV) (Severe acute re...)
Wichita State University

Curated by ChEMBL
LigandPNGBDBM50458462(CHEMBL4214066)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of SARS coronavirus 3CL protease using Dabcyl-KTSAVLQ/SGFRKME-Edans as substrate incubated for 30 mins followed by substrate addition meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed