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Found 4 Enz. Inhib. hit(s) with Target = 'Reverse transcriptase' and Ligand = 'BDBM50138406'
TargetReverse transcriptase(Human immunodeficiency virus 1)
Idenix An Msd

Curated by ChEMBL
LigandPNGBDBM50138406(3TC Triphosphate | CHEMBL1230 | LAMIVUDINE | Lamiv...)
Affinity DataIC50:  15nMAssay Description:Inhibition of full-length wild-type HIV1 reverse transcriptase expressed in Escherichia coli BL21(DE3) pre-incubated for 30 mins before addition of t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Idenix An Msd

Curated by ChEMBL
LigandPNGBDBM50138406(3TC Triphosphate | CHEMBL1230 | LAMIVUDINE | Lamiv...)
Affinity DataKd:  370nMAssay Description:Binding affinity to wild type HIV1 LAI reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Idenix An Msd

Curated by ChEMBL
LigandPNGBDBM50138406(3TC Triphosphate | CHEMBL1230 | LAMIVUDINE | Lamiv...)
Affinity DataKd:  130nMAssay Description:Binding affinity to HIV1 reverse transcriptase assessed as L-3'-azido-NTP incorporation in nascent DNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Idenix An Msd

Curated by ChEMBL
LigandPNGBDBM50138406(3TC Triphosphate | CHEMBL1230 | LAMIVUDINE | Lamiv...)
Affinity DataKd:  370nMAssay Description:Binding affinity to HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed