Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase LATS1' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase LATS1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 12.8nMAssay Description:Inhibition of human LATS1 using KKRNRRLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase LATS1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 13.3nMAssay Description:Inhibition of human LATS1 using KKRNRRLSVA as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase LATS1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding constant for LATS1 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase LATS1(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 42nMAssay Description:Binding constant for LATS1 kinase domainMore data for this Ligand-Target Pair