Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase tousled-like 2' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase tousled-like 2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human TLK2 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human TLK2 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for TLK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase tousled-like 2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for TLK2 kinase domainMore data for this Ligand-Target Pair