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Found 9 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM22397'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  10.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]WIN 35428 from human DAT transiently expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  13.4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  27.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  31.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wake Forest University

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM22397(WIN 35,428 | [3H]WIN 35,428 | methyl (1R,2S,3S,5S)...)
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed