Found 31 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50005548'
Affinity DataKi: 10nMAssay Description:Inhibition of human recombinant DAT expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]WIN-from cocaine site of dopamine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Inhibition of DAT in rat synaptosomal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to dopamine transporter (DAT) using [3H]WIN-35428 as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of dopamine (DA) uptake into rat brain synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Binding affinity to DAT (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:Inhibition of the uptake of tritiated dopamine (DA) in rat synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of full-length recombinant human DAT expressed in CHOK1 cells assessed as reduction in [3H]dopamine uptake pretreated for 20 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]dopamine reuptake at human DAT expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of [3H]BTCP binding to the dopamine transporter.More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of [3H]dopamine uptake at the dopamine transporter.More data for this Ligand-Target Pair
Affinity DataIC50: 115nMAssay Description:Inhibition of [3H]BTCP binding to the dopamine transporter.More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of [3H]dopamine uptake at dopamine transporter.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of [3H]dopamine uptake at the dopamine transporter.More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamineMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of dopamine uptake at dopamine transporter.More data for this Ligand-Target Pair