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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent noradrenaline transporter' and Ligand = 'BDBM50202381'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences

Curated by ChEMBL
LigandPNGBDBM50202381((RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]pipero...)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]RTI-55 from human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences

Curated by ChEMBL
LigandPNGBDBM50202381((RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]pipero...)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]RTI-55 from human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences

Curated by ChEMBL
LigandPNGBDBM50202381((RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]pipero...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]NE uptake into human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Massachusetts College Of Pharmacy And Health Sciences

Curated by ChEMBL
LigandPNGBDBM50202381((RR/SS)-2-[1-(4-chlorophenyl)-3-methylbutyl]pipero...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]NE uptake into human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed